中文名称: | TPI-1 | ||||
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英文名称: | TPI-1 | ||||
别名: | 2',5'-二氯-[1,1'-联苯基]-2,5-二酮 2',5'-Dichloro-[1,1'-biphenyl]-2,5-dione | ||||
CAS No: | 79756-69-7 | 分子式: | C12H6Cl2O2 | 分子量: | 253.08 |
CAS No: | 79756-69-7 | ||||
分子式: | C12H6Cl2O2 | ||||
分子量: | 253.08 |
一种SHP-1的抑制剂;抑制重组SHP-1的IC50值为40nM。
TPI-1, also known as Tyrosine Phosphatase Inhibitor 1, is a SHP-1 inhibitor. TPI-1 selectively increased SHP-1 phospho-substrates (pLck-pY394, pZap70, and pSlp76) in Jurkat T cells but had little effects on pERK1/2 or pLck-pY505 regulated by phosphatases SHP-2 or CD45, respectively. TPI-1 induced mouse splenic-IFN-gamma(+) cells in vitro, approximately 58-fold more effective than sodium stibogluconate, and increased mouse splenic-pLck-pY394 and -IFN-gamma(+) cells in vivo.
本计算器可帮助您计算出特定溶液中溶质的质量、溶液浓度和体积之间的关系,公式为:
质量 (g) = 浓度 (mol/L) x 体积 (L) x 分子量 (g/mol)
摩尔浓度计算公式
用本工具协助配置特定浓度的溶液,使用的计算公式为:
开始浓度 x 开始体积 = 最终浓度 x 最终体积
稀释公式
稀释公式一般简略地表示为:C1V1 = C2V2 ( 输入 输出 )