2020-10-20

1: Leaver D, Cleary B, Nguyen NT, Priebbenow DL, Lagiakos HR, Sanchez J, Xue L, 
Huang F, Sun Y, Mujumdar P, Mudududdla R, Varghese S, Teguh S, Charman SA, White 
K, Katneni K, Cuellar M, Strasser J, Dahlin J, Walters MA, Street I, Monahan B, 
Jarman KE, Jousset Sabroux H, Falk H, Chung M, Hermans S, Parker MW, Thomas T, 
Baell JB. Discovery of benzoylsulfonohydrazides as potent inhibitors of the 
histone acetyltransferase KAT6A. J Med Chem. 2019 Jun 29. doi: 
10.1021/acs.jmedchem.9b00665. [Epub ahead of print] PubMed PMID: 31256587.

2: Baell JB, Leaver DJ, Hermans SJ, Kelly GL, Brennan MS, Downer NL, Nguyen N, 
Wichmann J, McRae HM, Yang Y, Cleary B, Lagiakos HR, Mieruszynski S, Pacini G, 
Vanyai HK, Bergamasco MI, May RE, Davey BK, Morgan KJ, Sealey AJ, Wang B, Zamudio 
N, Wilcox S, Garnham AL, Sheikh BN, Aubrey BJ, Doggett K, Chung MC, de Silva M, 
Bentley J, Pilling P, Hattarki M, Dolezal O, Dennis ML, Falk H, Ren B, Charman 
SA, White KL, Rautela J, Newbold A, Hawkins ED, Johnstone RW, Huntington ND, Peat 
TS, Heath JK, Strasser A, Parker MW, Smyth GK, Street IP, Monahan BJ, Voss AK, 
Thomas T. Inhibitors of histone acetyltransferases KAT6A/B induce senescence and 
arrest tumour growth. Nature. 2018 Aug;560(7717):253-257. doi: 
10.1038/s41586-018-0387-5. Epub 2018 Aug 1. PubMed PMID: 30069049.